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Re: Digest Number 112

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You won't be able to maintain an erection; you will gain weight, and the

more weight you gain, the worse your diabetes will get; you will go blind;

your digestive system will quit working (gastroparesis), which will make

your diabetes control worse, and you will end up eating basically bland

baby food; your body parts will get amputated, a little bit at a time

(surgeons call it " slice and dice " ). It will start with your toes, then

your feet, then your lower legs. But first you will go through numerous

procedures because of sores that won't heal, etc. And you will be numb from

your waist down. And you will have trouble walking. And you will get cracks

on your heels and other sores on your feet and lower limbs that absolutely

will not heal. And you will take many different pills, and be hospitalized

numerous times. And you will be denied insurance. And you won't be able to

find work. And you will apply for welfare, but you will be turned down

because they will tell you you can still work. But none of the jobs that

offer medical insurance will hire you because you are such a high risk. And

you will be poor. And you will be depressed.

And you will get gangrene. And you will go blind. And your blood pressure

will skyrocket (more pills). And you will have a heart attack or two. And

then you will die.

HAVE A NICE DAY!

-In The Rapid Exchange of Information, Grammar, Spelling & Proper Sentence

Structure Are Low On My Priority List.- PK

PAUL KOSSART Peru, IL USA

NMRA, LDSIG, OPSIG, BRHS, TP & W-HS

LaSalle & Bureau County Model R.R. Club

Chicago, Burlington & Quincy Model R.R. (HO-1969)

" Serving Agriculture & Industry In The Illiniwek River Valley "

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Ahhh... Pleasant dreams everyone! G'nite!

/Celine Kossart wrote:

>

>

> You won't be able to maintain an erection; you will gain weight, and the

> more weight you gain, the worse your diabetes will get; you will go blind;

> your digestive system will quit working (gastroparesis), which will make

> your diabetes control worse, and you will end up eating basically bland

> baby food; your body parts will get amputated, a little bit at a time

> (surgeons call it " slice and dice " ). It will start with your toes, then

> your feet, then your lower legs. But first you will go through numerous

> procedures because of sores that won't heal, etc. And you will be numb from

> your waist down. And you will have trouble walking. And you will get cracks

> on your heels and other sores on your feet and lower limbs that absolutely

> will not heal. And you will take many different pills, and be hospitalized

> numerous times. And you will be denied insurance. And you won't be able to

> find work. And you will apply for welfare, but you will be turned down

> because they will tell you you can still work. But none of the jobs that

> offer medical insurance will hire you because you are such a high risk. And

> you will be poor. And you will be depressed.

>

> And you will get gangrene. And you will go blind. And your blood pressure

> will skyrocket (more pills). And you will have a heart attack or two. And

> then you will die.

>

> HAVE A NICE DAY!

>

> -In The Rapid Exchange of Information, Grammar, Spelling & Proper Sentence

> Structure Are Low On My Priority List.- PK

>

> PAUL KOSSART Peru, IL USA

> NMRA, LDSIG, OPSIG, BRHS, TP & W-HS

> LaSalle & Bureau County Model R.R. Club

> Chicago, Burlington & Quincy Model R.R. (HO-1969)

> " Serving Agriculture & Industry In The Illiniwek River Valley "

>

> ------------------------------------------------------------------------

> Did you know that ONElist hosts some of the largest lists on the Internet?

> http://www.ONElist.com

> Our scaleable system is the most reliable free e-mail service on the Internet!

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I wrote to Roy Dahl:

<< ... And you will get gangrene. And you will go blind. And your blood

pressure will skyrocket (more pills). And you will have a heart attack or

two. And then you will die. >>

And Kossart replied:

<< HAVE A NICE DAY! >>

" Other than *that*, Mrs. Lincoln, did you enjoy the play? "

Susie ;D

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Did I miss something? Why was this posted? I know I have been quite for

awhile but have had alot to do. This just surprised me.

Stormy

Re: Digest Number 112

>

>

>

>You won't be able to maintain an erection; you will gain weight, and the

>more weight you gain, the worse your diabetes will get; you will go blind;

>your digestive system will quit working (gastroparesis), which will make

>your diabetes control worse, and you will end up eating basically bland

>baby food; your body parts will get amputated, a little bit at a time

>(surgeons call it " slice and dice " ). It will start with your toes, then

>your feet, then your lower legs. But first you will go through numerous

>procedures because of sores that won't heal, etc. And you will be numb from

>your waist down. And you will have trouble walking. And you will get cracks

>on your heels and other sores on your feet and lower limbs that absolutely

>will not heal. And you will take many different pills, and be hospitalized

>numerous times. And you will be denied insurance. And you won't be able to

>find work. And you will apply for welfare, but you will be turned down

>because they will tell you you can still work. But none of the jobs that

>offer medical insurance will hire you because you are such a high risk. And

>you will be poor. And you will be depressed.

>

>And you will get gangrene. And you will go blind. And your blood pressure

>will skyrocket (more pills). And you will have a heart attack or two. And

>then you will die.

>

>

>HAVE A NICE DAY!

>

>

>

>-In The Rapid Exchange of Information, Grammar, Spelling & Proper Sentence

>Structure Are Low On My Priority List.- PK

>

>PAUL KOSSART Peru, IL USA

>NMRA, LDSIG, OPSIG, BRHS, TP & W-HS

>LaSalle & Bureau County Model R.R. Club

>Chicago, Burlington & Quincy Model R.R. (HO-1969)

> " Serving Agriculture & Industry In The Illiniwek River Valley "

>

>------------------------------------------------------------------------

>Did you know that ONElist hosts some of the largest lists on the Internet?

>http://www.ONElist.com

>Our scaleable system is the most reliable free e-mail service on the

Internet!

>

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Stormy writes:

<< Did I miss something? Why was this posted? I know I have been quite for

awhile but have had alot to do. This just surprised me. >>

Our new member Roy Dahl wrote in ... Here, I'll let him tell you ...

<< ... In August, 1996 I suffered from the same symptoms and again saw the

family doctor who again, indicated I was certainly diabetic. Since then, I

have made some adjustments, but consider myself a " bad diabetic " , in that I

don't follow the rules very well. Most days, my blood sugar drifts between

10.0 - 22.0 (normal is supposed to be between 4 - 8). I still indulge in a

dessert at supper, and every now and then, will enjoy a coke or a chocolate

bar. I know, I know - I'm not supposed to be doing these things! How do I

stop? ... >>

I was presenting a dire scenario to Roy, hoping it would help motivate him.

Susie

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oh ok. I was just surprised by the post. It does make you think though. My

new ALT came back 125. I don't know what is wrong I have to go every week to

get these done. From what I understand they are suppose to be between 5-40

whatever. I don't know how this works. Getting frustrated. I still feel

pretty good. I have been spending time with the kids. They don't know what

to do with me. They are use to me being so sick that I didn't really PLAY

with them. I went outside yesterday with my youngest that has this water

balloon ball that is on two strings and you both have to pull on the 2

strings to get it to the other person and hope the balloon pops on the

other. She thought it was great. I haven't been able to do stuff like that

for sooooooooo long. BTW I got wet. She really loved that one.

Take care all.

Stormy

Re: Digest Number 112

>From: OtterCritter@...

>

>Stormy writes:

>

><< Did I miss something? Why was this posted? I know I have been quite for

>awhile but have had alot to do. This just surprised me. >>

>

>Our new member Roy Dahl wrote in ... Here, I'll let him tell you ...

>

><< ... In August, 1996 I suffered from the same symptoms and again saw the

>family doctor who again, indicated I was certainly diabetic. Since then, I

>have made some adjustments, but consider myself a " bad diabetic " , in that I

>don't follow the rules very well. Most days, my blood sugar drifts between

>10.0 - 22.0 (normal is supposed to be between 4 - 8). I still indulge in a

>dessert at supper, and every now and then, will enjoy a coke or a chocolate

>bar. I know, I know - I'm not supposed to be doing these things! How do I

>stop? ... >>

>

>I was presenting a dire scenario to Roy, hoping it would help motivate him.

>

>Susie

>

>

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Stormy reports still having elevated ALT numbers on her most recent liver

test. Here is a message from a professor to his students, taken from the

web:

<< From: Dr Velan -- Date: 5/22/97

To simplify matters, there are only three true tests of hepatocyte function,

and one of them doesn't even come under the banner of " liver function

tests " !

The best test of medium to long-term hepatic function is serum albumin

(although liver disease is not the only cause of hypoalbuminaemia - e.g.

nephrotic syndrome and protein malnutrition). Albumin is synthesised at a

rate of 12 g/day, making up half of all hepatic protein synthesis. The

half-life of albumin in the circulation is 17 to 20 days, hence impaired

synthesis may take months to become apparent.

The best test of short-term hepatic function is the prothrombin time (not

usually included in " LFTs " ), which tests the integrity of the extrinsic

coagulation cascade - clotting factors II, VII, IX & X are produced in the

liver and have short half-lives. Acute liver dysfunction typically induces a

prolonged prothrombin time which is not corrected by administration of

Vitamin K. Bleeding from the GIT is a common cause of death in patients with

fulminant hepatic failure.

Serum bilirubin is a much less sensitive test of hepatic function, and may

be normal in compensated cirrhosis or early in the course of fulminant

hepatic failure. The serum bilirubin is more sensitive to cholestasis than

to hepatocyte dysfunction.

The other " liver function tests " (ALP, GGT, ALT, AST) measure enzyme levels

which reflect ongoing hepatic inflammation, necrosis and/or cholestasis,

rather than hepatocyte function. >>

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Someone needs to say it every once in a while to keep us all motivated,

Stormy. Nothing to take exception to.

Winston

Re: Digest Number 112

>

>

>>

>>

>>

>>You won't be able to maintain an erection; you will gain weight, and the

>>more weight you gain, the worse your diabetes will get; you will go blind;

>>your digestive system will quit working (gastroparesis), which will make

>>your diabetes control worse, and you will end up eating basically bland

>>baby food; your body parts will get amputated, a little bit at a time

>>(surgeons call it " slice and dice " ). It will start with your toes, then

>>your feet, then your lower legs. But first you will go through numerous

>>procedures because of sores that won't heal, etc. And you will be numb

from

>>your waist down. And you will have trouble walking. And you will get

cracks

>>on your heels and other sores on your feet and lower limbs that absolutely

>>will not heal. And you will take many different pills, and be hospitalized

>>numerous times. And you will be denied insurance. And you won't be able to

>>find work. And you will apply for welfare, but you will be turned down

>>because they will tell you you can still work. But none of the jobs that

>>offer medical insurance will hire you because you are such a high risk.

And

>>you will be poor. And you will be depressed.

>>

>>And you will get gangrene. And you will go blind. And your blood pressure

>>will skyrocket (more pills). And you will have a heart attack or two. And

>>then you will die.

>>

>>

>>HAVE A NICE DAY!

>>

>>

>>

>>-In The Rapid Exchange of Information, Grammar, Spelling & Proper Sentence

>>Structure Are Low On My Priority List.- PK

>>

>>PAUL KOSSART Peru, IL USA

>>NMRA, LDSIG, OPSIG, BRHS, TP & W-HS

>>LaSalle & Bureau County Model R.R. Club

>>Chicago, Burlington & Quincy Model R.R. (HO-1969)

>> " Serving Agriculture & Industry In The Illiniwek River Valley "

>>

>>------------------------------------------------------------------------

>>Did you know that ONElist hosts some of the largest lists on the Internet?

>>http://www.ONElist.com

>>Our scaleable system is the most reliable free e-mail service on the

>Internet!

>>

>

>

>------------------------------------------------------------------------

>Looking for the perfect gift for a friend?

>http://www.ONElist.com

>Tell them about ONElist's 115,000 free e-mail communities!

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Thank you for the information. I printed it up and I am going to take it

with me this week when I go back to the DR. Like I said I feel ok and have

more energy than I have had in years. So I am not letting it get me down. I

am having too much fun.

Hugs

Stormy

Re: Digest Number 112

>From: OtterCritter@...

>

>Stormy reports still having elevated ALT numbers on her most recent liver

>test. Here is a message from a professor to his students, taken from the

>web:

>

><< From: Dr Velan -- Date: 5/22/97

>

>To simplify matters, there are only three true tests of hepatocyte

function,

>and one of them doesn't even come under the banner of " liver function

>tests " !

>

>The best test of medium to long-term hepatic function is serum albumin

>(although liver disease is not the only cause of hypoalbuminaemia - e.g.

>nephrotic syndrome and protein malnutrition). Albumin is synthesised at a

>rate of 12 g/day, making up half of all hepatic protein synthesis. The

>half-life of albumin in the circulation is 17 to 20 days, hence impaired

>synthesis may take months to become apparent.

>

>The best test of short-term hepatic function is the prothrombin time (not

>usually included in " LFTs " ), which tests the integrity of the extrinsic

>coagulation cascade - clotting factors II, VII, IX & X are produced in the

>liver and have short half-lives. Acute liver dysfunction typically induces

a

>prolonged prothrombin time which is not corrected by administration of

>Vitamin K. Bleeding from the GIT is a common cause of death in patients

with

>fulminant hepatic failure.

>

>Serum bilirubin is a much less sensitive test of hepatic function, and may

>be normal in compensated cirrhosis or early in the course of fulminant

>hepatic failure. The serum bilirubin is more sensitive to cholestasis than

>to hepatocyte dysfunction.

>

>The other " liver function tests " (ALP, GGT, ALT, AST) measure enzyme levels

>which reflect ongoing hepatic inflammation, necrosis and/or cholestasis,

>rather than hepatocyte function. >>

>

>

>

>------------------------------------------------------------------------

>Have you visited the new ONElist home page lately?

>http://www.ONElist.com

>ONElist: The Leading e-mail list and community service on the Internet!

>

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Guest guest

,

Thanks for this posting. I sometimes get depressed and say, " The hell with

it. " I have printed your post and will use it to remind myself of the

consequences of such an attitude.

Thanks again.

Mr. Edd

None of us is as smart as all of us.

Re: Digest Number 112

>>

>>

>>>

>>>

>>>

>>>You won't be able to maintain an erection; you will gain weight, and the

>>>more weight you gain, the worse your diabetes will get; you will go

blind;

>>>your digestive system will quit working (gastroparesis), which will make

>>>your diabetes control worse, and you will end up eating basically bland

>>>baby food; your body parts will get amputated, a little bit at a time

>>>(surgeons call it " slice and dice " ). It will start with your toes, then

>>>your feet, then your lower legs. But first you will go through numerous

>>>procedures because of sores that won't heal, etc. And you will be numb

>from

>>>your waist down. And you will have trouble walking. And you will get

>cracks

>>>on your heels and other sores on your feet and lower limbs that

absolutely

>>>will not heal. And you will take many different pills, and be

hospitalized

>>>numerous times. And you will be denied insurance. And you won't be able

to

>>>find work. And you will apply for welfare, but you will be turned down

>>>because they will tell you you can still work. But none of the jobs that

>>>offer medical insurance will hire you because you are such a high risk.

>And

>>>you will be poor. And you will be depressed.

>>>

>>>And you will get gangrene. And you will go blind. And your blood pressure

>>>will skyrocket (more pills). And you will have a heart attack or two. And

>>>then you will die.

>>>

>>>

>>>HAVE A NICE DAY!

>>>

>>>

>>>

>>>-In The Rapid Exchange of Information, Grammar, Spelling & Proper

Sentence

>>>Structure Are Low On My Priority List.- PK

>>>

>>>PAUL KOSSART Peru, IL USA

>>>NMRA, LDSIG, OPSIG, BRHS, TP & W-HS

>>>LaSalle & Bureau County Model R.R. Club

>>>Chicago, Burlington & Quincy Model R.R. (HO-1969)

>>> " Serving Agriculture & Industry In The Illiniwek River Valley "

>>>

>>>------------------------------------------------------------------------

>>>Did you know that ONElist hosts some of the largest lists on the

Internet?

>>>http://www.ONElist.com

>>>Our scaleable system is the most reliable free e-mail service on the

>>Internet!

>>>

>>

>>

>>------------------------------------------------------------------------

>>Looking for the perfect gift for a friend?

>>http://www.ONElist.com

>>Tell them about ONElist's 115,000 free e-mail communities!

>

>

>------------------------------------------------------------------------

>Did you know that knowledge is power?

>http://www.ONElist.com

>Join a new ONElist e-mail community and strengthen your mind!

>

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In a message dated 99-04-12 00:19:08 EDT, you write:

<< And then you will die. >>

PAUL: YOU SAID IT LIKE IT IS! ONE HAS TO GET CONTROL OF HIS BLOOD SUGAR

LEVELS! AND

God's Speed.

***Robin***

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ALT is one of the liver function test. I can't really explain it because I

am still learning myself. I think one of the other people could probably

explain it better.

Stormy

Re: Digest Number 112

>From: Om8421@...

>

>Dear Stormy,

> what does Alt mean....still learning here.....Merry

>

>------------------------------------------------------------------------

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http://www.mtio.com/mclfa/lfalt1.htm

http://www.hepplace.com/alt.html

Re: Digest Number 112

>

>

>>From: Om8421@...

>>

>>Dear Stormy,

>> what does Alt mean....still learning here.....Merry

>>

>>------------------------------------------------------------------------

>>Share the wealth!

>>http://www.ONElist.com

>>Tell a friend about ONElist's 115,000 free e-mail communities!

>>

>

>

>------------------------------------------------------------------------

>

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In a message dated 99-04-14 22:53:09 EDT, you write:

<< Hi everyone I have been taking Rezulen for about a year now it has

really helped with my blood sugars. I just had the liver tests my Dr.

said I should keep taking it for now. I take 400mg a day. I would like

to hear from you all >>

KATHIE: I have been on 400mg of Rezulin since September of 98. My blood

sugars have really dropped (from over 200mg/dl to under 120mg/dl). I take

monthly liver test and so far no damage to my liver. I pray that it

continues to help my blood sugar levels and not damage the liver. AND

God's Speed.

***Robin***

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Hi everyone I have been taking Rezulen for about a year now it has

really helped with my blood sugars. I just had the liver tests my Dr.

said I should keep taking it for now. I take 400mg a day. I would like

to hear from you all.kathie

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Hi Kathie,

My doctor started me out on 400 mg. daily of Rezulin, then increased to 300

mg. twice daily and later decreased to 300 mg. once daily. Reduction was

because I have a problem with water retention and that is a side effect of

Rezulin. Do you also take insulin? I take a small amount twice daily and

it really boosts the effects of the insulin. Only once my liver enzymes

were elevated and he repeated them in two weeks and considered taking me

off the medicine but didn't as the second set of liver tests were normal.

Rezulin is in the news quite a lot and sometimes I am a little scared to

take it.

I took Redux and it worked wonderfully well for me and I was really sad

they took it off the market. I know someone who took Duract for pain and

almost died and has unreversible liver damage. She is a single Mom with 3

kids, the youngest in 1st grade and I really feel for her.

Sorry to be so long winded but am glad you brought up the subject of

Rezulin.

If you wish, you can e-mail me privately so we won't bore the others on the

list to death!

Kay

To: diabetes_intonelist

Subject: Re: Digest Number 112

Date: Wednesday, April 14, 1999 9:00 PM

Hi everyone I have been taking Rezulen for about a year now it has

really helped with my blood sugars. I just had the liver tests my Dr.

said I should keep taking it for now. I take 400mg a day. I would like

to hear from you all.kathie

------------------------------------------------------------------------

Did you know that ONElist hosts some of the largest lists on the Internet?

http://www.ONElist.com

Our scaleable system is the most reliable free e-mail service on the

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Believe me it MOTIVATED me. I wasn't upset about the post. I thought maybe

someone had something really terrible happen to them.

Stormy

Re: Digest Number 112

>>

>>

>>>

>>>

>>>

>>>You won't be able to maintain an erection; you will gain weight, and the

>>>more weight you gain, the worse your diabetes will get; you will go

blind;

>>>your digestive system will quit working (gastroparesis), which will make

>>>your diabetes control worse, and you will end up eating basically bland

>>>baby food; your body parts will get amputated, a little bit at a time

>>>(surgeons call it " slice and dice " ). It will start with your toes, then

>>>your feet, then your lower legs. But first you will go through numerous

>>>procedures because of sores that won't heal, etc. And you will be numb

>from

>>>your waist down. And you will have trouble walking. And you will get

>cracks

>>>on your heels and other sores on your feet and lower limbs that

absolutely

>>>will not heal. And you will take many different pills, and be

hospitalized

>>>numerous times. And you will be denied insurance. And you won't be able

to

>>>find work. And you will apply for welfare, but you will be turned down

>>>because they will tell you you can still work. But none of the jobs that

>>>offer medical insurance will hire you because you are such a high risk.

>And

>>>you will be poor. And you will be depressed.

>>>

>>>And you will get gangrene. And you will go blind. And your blood pressure

>>>will skyrocket (more pills). And you will have a heart attack or two. And

>>>then you will die.

>>>

>>>

>>>HAVE A NICE DAY!

>>>

>>>

>>>

>>>-In The Rapid Exchange of Information, Grammar, Spelling & Proper

Sentence

>>>Structure Are Low On My Priority List.- PK

>>>

>>>PAUL KOSSART Peru, IL USA

>>>NMRA, LDSIG, OPSIG, BRHS, TP & W-HS

>>>LaSalle & Bureau County Model R.R. Club

>>>Chicago, Burlington & Quincy Model R.R. (HO-1969)

>>> " Serving Agriculture & Industry In The Illiniwek River Valley "

>>>

>>>------------------------------------------------------------------------

>>>Did you know that ONElist hosts some of the largest lists on the

Internet?

>>>http://www.ONElist.com

>>>Our scaleable system is the most reliable free e-mail service on the

>>Internet!

>>>

>>

>>

>>------------------------------------------------------------------------

>>Looking for the perfect gift for a friend?

>>http://www.ONElist.com

>>Tell them about ONElist's 115,000 free e-mail communities!

>

>

>------------------------------------------------------------------------

>Did you know that knowledge is power?

>http://www.ONElist.com

>Join a new ONElist e-mail community and strengthen your mind!

>

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Guest guest

I just don't understand why T2 goes faster than the speed of light at times.

Now that they took me off the Rezulin my blood sugars are going up real high

then down real low again. That does not do well with me. I feel like I am a

rollercoaster from you know where. I know that I am whining but I am just

frustrated right now. Sorry I will try to get in a better mood. Thanks.

Stormy

Re: Digest Number 112

>

>

>> <<< The ADA has issued guidelines to doctors that all adults 45 and

older

>> should receive annual testing for fasting blood glucose levels. This

should

>> go a long way toward locating the undiagnosed ones.>>>

>

>Hi Stormy,

>

>My doctor checked me about 6 weeks before I was diagnosed and I had a

fasting BG

>of 146 so he wanted to check it again in 3 months... Unfortunately my T-2

was

>catching up with me faster than that.

>

>

>

>

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Stormy writes:

<< ... Now that they took me off the Rezulin my blood sugars are going up

real high then down real low again. That does not do well with me. I feel

like I am a rollercoaster from you know where ... >>

Stormy and others, Rick Mendosa is a writer with diabetes expertise whose

web sites contain a wealth of information. His home page is

http://www.mendosa.com/ Here is an article he wrote regarding diabetes

medications (http://www.mendosa.com/newdrugs.htm):

Beyond Sulfonylureas -- The New Drugs for Blood Glucose Control

By Rick Mendosa

Life is getting more complicated for people with type 2 diabetes and the

doctors who treat them. But that's good. If you think you and your doctor

have a lot of glucose-lowering drugs to choose from now, hang onto your hat

as we look at what the biotech companies are developing. Until 1995, the

sulfonylurea class of drugs was the only choice other than insulin for

treating type 2 diabetes. Certainly you had a choice of brand, but they all

work the same way, by squeezing more insulin out of your beta cells and

improving insulin's ability to get glucose into the rest of your body.

Sulfonylurea drugs include Glucotrol (glipizide) and DiaBeta, Glynase, and

Micronase (glyburide).

The explosion of drugs available for controlling blood glucose began when

Glucophage (metformin) became available in 1995, quickly followed by Precose

(acarbose). Bristol-Myers Squibb's Glucophage works differently from the

sulfonylureas by keeping the liver from making too much sugar. Bayer

Corporation's Precose, a third class of drugs, slows carbohydrate digestion.

The fourth choice hit the market a year ago. Parke-'s Rezulin

(troglitazone) makes the body more sensitive to its insulin. In spite of

reports of liver damage in some people, the drug continues to be available

here with warnings that people who use it need very frequent liver tests.

Rezulin remains on the market here because it works well for most folks. In

one study, average levels of HbA1c dropped 1.4 percent. For example, if you

have an HbA1c level of 8, you might expect it to come down to 6.4.

Rezulin works even better in combination with a sulfonylurea. In fact, " Any

one of these drugs can be used in combination with any other, " says Dr.

W. Quick, a board-certified endocrinologist practicing near Kansas

City. " The research studies are a bit stronger for some of the combinations

than they are for others, but out here in clinical practice we use all the

combinations. "

" Vegetable soup " is what Dr. Quick calls the choices open to him and his

type 2 patients. " We can add any of several different ingredients and come

up with a slightly a slightly different flavor for individualized therapy

with the drugs that are available now. I am very impressed that we are doing

a heck of a lot better than we did in the past when we had just one flavor

to our soup. "

PRANDIN

Now, a fifth class of drugs hit the market in April, when Novo Nordisk and

Schering-Plough jointly launched Prandin (regaglinide). It works by

stimulating insulin secretion from the beta cells and differs from earlier

drugs both in its structure and how it is eliminated. It needs to be taken

just before each meal because it is so fast-acting.

Prandin may be even more effective than Rezulin. It reduced HbA1c levels by

2.1 percent in one study reported in the package insert that will come with

the drug.

Beyond Prandin, there is an explosion of research on glucose control drugs.

" As someone who has had diabetes for 48 years, I don't think that I have

ever seen a more exciting time, " says Dr. , associate dean and

professor of pharmacy practice at Washington State University College of

Pharmacy and a Certified Diabetes Educator.

ERGOSET

The glucose control drug probably closest to market after Prandin is

Ergoset. The FDA is considering its approval after receiving a New Drug

Application from its manufacturer, Ergo Science Corporation, in October.

" We are probably looking at an early 1999 launch, " says Donna LaVoie, Ergo

Science's executive director, corporate communications and investor

relations. & will market Ergoset under the terms of a

multimillion dollar deal the two companies signed this February.

Ergoset is a low-dose and fast-acting formulation of bromocriptine, which

doctors have prescribed for years in a different form to treat Parkinson's

disease. Unlike other diabetes control drugs that work at the gut level,

Ergoset's action is through the brain, resetting the body's clock that

regulates daily metabolic activity.

Studies of Ergoset show an average drop in HbA1c of 1.04 percent. But unlike

other studies, that's a measure only of the patients who responded well to

it, excluding the 36 percent who didn't.

The drug also has a lipid-lowering effect and is in Phase II trials for

obesity. And that's another problem in understanding its effectiveness.

Since patients on Ergoset lose weight, there's a question whether it lowers

HbA1c directly or because of weight loss, says Dr. Dan Baker, director of

drug information at Washington State University in Spokane.

" It is an interesting product, and it will be useful, " he believes. He notes

that two other weight-control drugs close to market may also help people

with diabetes reduce their blood glucose, Meridia and Xenical (see following

table).

TARGRETIN

Like Ergoset, Targretin's original target was another disease. And like Ergo

Science, Targretin's developer has a powerful corporate alliance that is

some indication of the likelihood the drug will actually come to market.

Ligand Pharmaceuticals developed Targretin to fight certain cancers, but

serendipitously discovered that it is also an insulin sensitizer. Ligand has

licensed marketing rights to Eli Lilly and Company for $99 million.

" Targretin is a Vitamin A derivative, " says Henry Niman, an associate

professor in the University of Pittsburgh's epidemiology department and the

scientific founder of Ligand's parent company.

The drug is in phase II trials for diabetes and probably won't be on the

market until three to four years from now, he says. " In animals it worked

great. It was as effective as one of the second generation compounds in

Rezulin's class, which are even more effective than Rezulin itself. " It also

reduced triglyceride levels.

BRL 49653

The second generation compound Dr. Niman is talking about is BRL 49653.

Kline Beecham, which developed the drug says that it is an insulin

sensitizer and is in Phase III trials.

Beyond that, the company releases little additional information. " It's

frustrating to us in pharmacy and in medicine to project what is going to

happen in the future with drug therapy, " Dr. says. " For almost

every new drug that comes out there is almost nothing in the scientific

literature until about the time the FDA recommends it for approval. "

SP-134101

Among all the other drugs now in clinical and preclinical trials to reduce

blood glucose levels perhaps the most interesting is SP-134101, which Shaman

Pharmaceuticals is developing. The drug just started Phase I trials and

probably won't hit the market until about 2003, according to Vice President

J. D. Haldeman.

What makes SP-134101 exciting is that it is the first of 21 compounds the

company found in tropical plants that lower blood glucose levels in animal

models. " SP-134101 comes from a plant that grows in the southeastern part of

the U.S. and Mexico, " she says. " We will be isolating it directly from the

plant. "

DRUG PROBLEMS

Even if all of these drugs prove effective in reducing blood glucose, that's

not the end of the story. " I consider effectiveness as only a minor factor

in my decision-making, " Dr. Quick says. " Other factors to consider include

cost, side effects, rules about time of administration, taste and other

eccentricities of the pill, and contraindications. "

He emphasizes that these issues affect how well patients use these drugs.

And as Dr. points out, little of this information will be available

until just before they come on the market. Stay tuned.

An edited version of this article appeared as " Beyond Sulfonylureas " in

Diabetes Wellness Letter, May 1998, pages 1-4.

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  • 2 years later...
Guest guest

Hi Debbie, My name is Sharon and I went to Curlin in Sept of 99. Bad mistake

! I am now getting ready to go to Dr.L. Out of all of the doctors I have

talked to I believe for him to be the very best choice.(MY OPINION)I live in

Raleigh 30 mins from Dr Berger but have chose to go to Dr L. I love the fact

that he does'nt think twice about answering my phone calls or emails. And he

has always been very honest with me. With Curlin I know that you are out of

$500.00 but it could be worst. I am out of the whole thing and now I am

going to pay another$5,500.00 but I believe tit to be wirth it this time.

Stick with your gut feelings. If I would have went with mine when I went to

Curlin's office I would have gotten up walked out and came right back to NC

without him touching me. Again my opinion. Sharon

Digest Number 112

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