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This is from Medscape

sorry if you can't read the charts

Human Dermal Safety Studies with Eflornithine HCl 13.9% Cream (VaniqaTM), a

Novel Treatment for Excessive Facial Hair

Janet G. Hickman, Education and Research Foundation Inc., Lynchburg, VA

24501, USA; Ferdinand Huber and Palmisano, Bristol Myers Squibb,

Princeton, NJ 08540, USA.

[Current Medical Research and Opinion 16(4):235-244, 2001]

Summary

Eflornithine HCl 13.9% cream (VaniqaTM) is a novel treatment for the

management of unwanted facial hair in women. This paper reports the results

of four modified open-label, within-subject vehicle-controlled studies

evaluating the dermal safety of this topical treatment. In a repeated insult

patch test (230 subjects), erythema with oedema occurred in 38.9% of

subjects treated with eflornithine HCl 13.9% cream and 4.8% of subjects

treated with vehicle cream. Challenge applications at previously untested

sites following the three-week induction period produced noticeable erythema

or greater on only four sites treated with eflornithine HCl 13.9% cream and

one vehicle-treated site. The erythema at these sites subsided substantially

within 24 hours. In a three-week cumulative irritation study (30 subjects),

the mean irritation score for sites treated with eflornithine HCl 13.9%

cream was 1.33, compared with 0.76 at vehicle-treated sites and 3.09 at

positive-control (sodium lauryl sulphate-treated) sites (p < 0.001 between

all three groups). In a phototoxicity study (25 subjects), irradiated sites

showed either no reaction (40% of both sites treated with eflornithine HCl

13.9% cream and vehicle-treated sites), or mild erythema subsiding in all

cases but one within 24 hours. No reaction was seen at non-irradiated sites.

In a photocontact allergy study (30 subjects), challenge with eflornithine

HCl 13.9% cream or its vehicle alone produced either no reaction or mild

erythema subsiding within 24 hours at both irradiated and non-irradiated

sites. No serious adverse events were reported during the studies, and the

only adverse events considered related to treatment were pruritus (three

subjects) and dry skin at test site (one subject). These results demonstrate

that eflornithine HCl 13.9% cream does not have contact sensitising,

photocontact allergic or phototoxic properties. It can cause irritation

under exaggerated conditions of use. Eflornithine HCl 13.9% cream,

therefore, has a favourable dermal safety profile appropriate for a topical

treatment to be applied routinely.

Introduction

Many women who suffer from unwanted facial hair regard this as a defect in

their appearance. This can lead to psychosocial problems ranging from

withdrawal from social situations to anxiety and depression.[1-3]

Until recently, there has been no proven safe and effective topical

medication for controlling facial hair growth. Popular methods for removing

facial hair include shaving, plucking (tweezing), waxing, chemical

depilation and electrolysis.[4-6] These methods are often painful,

inconvenient or expensive. Therefore a treatment that reduces the need for

hair removal would bring benefits to women with unwanted facial hair.

Eflornithine HCl 13.9% cream (VaniqaTM) is a convenient topical treatment

for reducing facial hair growth. Eflornithine is an irreversible inhibitor

of ornithine decarboxylase, an enzyme responsible for the catalysis of

ornithine to putrescine.[7] Putrescine and other polyamines play an

important role in the regulation of cell growth and differentiation.[8]

Ornithine decarboxylase is present in the hair follicle and studies in

animal models have shown that eflornithine is a potent inhibitor of hair

growth.[9] Clinical evaluation of eflornithine HCl 13.9% cream shows this

topical agent to be effective in reducing facial hair growth in women (Wolf

et al., manuscript in preparation).

Extensive preclinical evaluations have shown eflornithine HCl 13.9% cream to

have predictable pharmacokinetics and a favourable toxicological profile

(Shander and , personal communication). Clinical studies in humans

showed that eflornithine HCl 13.9% cream has a low percutaneous absorption

(< 1%) under conditions of likely clinical use, and that any absorbed

eflornithine is rapidly excreted in urine without being metabolised

(Malhotra, manuscript in preparation).

Dermal safety is an important consideration for a topical treatment that is

to be used regularly. This paper reports the results of four dermatological

studies in humans, which evaluated the potential of eflornithine HCl 13.9%

cream and its vehicle to cause contact sensitisation, irritation,

phototoxicity and photocontact allergy. The contact sensitisation and

cumulative irritation studies both involved exaggerated use of eflornithine

HCl 13.9% cream in that the cream was applied and maintained under occlusive

dressings for 21 days.

Contact Sensitisation Study

Subjects and Methods

In total, 230 healthy subjects were enrolled in a 37-day, modified,

open-label, single-centre, within-subject vehicle-controlled study, to

examine the contact sensitisation potential of topical treatment with

eflornithine HCl 13.9% cream and its vehicle alone. The study consisted of a

three-week induction period of exaggerated use under occlusive patches,

followed two weeks later by a single-dose challenge given at a previously

untested site (modified Draize skin sensitisation test). Skin responses to

challenge were used to assess contact sensitisation.[10-12]

Subjects were at least 18 years of age. Female subjects were sterile or had

a negative pregnancy test on entry into the study and agreed to use

contraception for the duration of the study. Subjects were not permitted to

use medications such as anti-histamines, corticosteroids, analgesics and

anti-inflammatories during the study.

Exclusion criteria were concomitant skin pathologies, atopic

dermatitis/eczema, psoriasis or asthma, a history of hypersensitivity to any

component of the formulations, treatment with medications such as

anti-histamines, corticosteroids, analgesics and anti-inflammatories in the

week before the study, treatment with investigational medicines during the

four weeks before the study, current pregnancy or nursing, a history of

pregnancy while using contraception, and skin pigmentation likely to

interfere with assessment of skin reactions.

Eflornithine HCl (2-(difluoromethyl)-D,L-ornithine monohydrochloride 13.9%

(w/w) cream, equivalent to 15% when expressed as the monohydrate) (VaniqaTM)

(0.2 g) was applied using a Hill Top Chamber under occlusive patches to a

site 1.8 cm in diameter on the upper back of each subject. Vehicle cream was

applied to a second site in the same manner. Patch test sites were selected

to avoid skin blemishes, moles, scars and the midline over the spine.

During the three-week induction period, doses of eflornithine HCl 13.9%

cream and vehicle were applied to the test site three times a week (Monday,

Wednesday and Friday) and left in place until the next application. During

the subsequent two-week rest period, no treatment was applied. This was

followed by application of single 48-hour challenge doses made at previously

untested skin sites.

Skin reactions were evaluated five minutes after each induction patch was

removed (three times a week for three weeks), and both five minutes and 24

hours after the challenge patches were removed, using a five-point ordinal

scale:

No sign of reaction

Slight erythema

Noticeable erythema with slight infiltration

Erythema with marked oedema

Erythema with oedema and blistering

If the test product produced a severe reaction (Grades 3 or 4), applications

were moved to a new skin site, or the subject was withdrawn from the study

if necessary.

Adverse events were recorded for the duration of the study for all subjects

enrolled.

Results

The demographic characteristics of the enrolled subjects are shown in Table

1. Two-hundred and eight of the 230 subjects enrolled completed the study

and 185 made all scheduled visits (22 subjects missed one scheduled visit

and one subject missed two scheduled visits). All 208 subjects were included

in the analysis. The remaining 22 subjects withdrew from the study

prematurely for the following reasons: 14 left of their own volition, four

were lost to follow-up, three missed two or more consecutive visits and one

withdrew owing to an adverse event not considered to be related to the study

therapy.

During the three-week induction period with eflornithine HCl 13.9% cream, 81

sites (38.9%) had response scores of 3 or 4. Of subjects completing the

study, five (2.4%) showed no evidence of reaction at test sites (Grade 0)

during induction with eflornithine HCl 13.9% cream. During induction with

vehicle cream alone, 203 sites (97.6%) had scores of 1 or greater on at

least one occasion, but only 10 sites (4.8%) scored 3 or 4.

Challenge with eflornithine HCl 13.9% cream produced either no reaction

(score of 0) or slight erythema (score of 1) on 98.1% of test sites

(204/208) (Table 2). Three sites had a score of 2 (noticeable erythema with

slight infiltration) five minutes after patch removal, falling to 1 or 0

within 24 hours, and 1 had a score of 4 (erythema with oedema and

blistering), which fell to 2 within 24 hours. After challenge with vehicle

only, all sites had a score of 0 or 1, with the exception of one score of 2,

which fell to 1 within 24 hours.

No serious adverse events were reported during the contact sensitisation

study. In total, 11 adverse events were reported in 10 subjects (4.3%):

headache (three subjects), pruritus (two subjects), accidental injury (one

subject), cyst (one subject), infection (one subject), back pain (one

subject), cholelithiasis (one subject), and diarrhoea (one subject). Of

these, only pruritus at patch sites (two subjects), occurring 10-15 days

into the study was considered related to treatment.

Cumulative Irritation Study

Subjects and Methods

In total, 30 healthy subjects were enrolled in an open-label, single-centre,

within-subject vehicle- and positive-controlled study to evaluate the

irritation potential of topical treatment with eflornithine HCl 13.9% cream,

its vehicle alone and a known irritant - sodium lauryl sulphate (0.5%) in

petrolatum. The study consisted of a three-week period of exaggerated use,

during which skin responses were assessed daily.[10-13] Subjects were

enrolled based on the same criteria as before.

Each subject received eflornithine HCl 13.9% cream, vehicle alone and 0.5%

(w/w) sodium lauryl sulphate in petrolatum (0.2 g of each), which were

applied under separate occlusive patches as described before. Each patch was

removed and fresh test materials were applied six days a week (Monday to

Saturday) for three weeks. The final patch was removed 48 hours after

application.

Cumulative irritation was measured five minutes after patch removal using a

five-point ordinal scale, as before. Once a score of 4 was observed, no

further applications of that treatment were made to the subject and a score

of 4 was assigned for the remainder of the study. Adverse events were

recorded for the duration of the study.

The statistical significance of the scores obtained was assessed using the

Friedman test. An approximation to the Friedman test was employed using the

procedure PROC GLM in SAS. This procedure was applied after a ranking was

performed within subject on the treatment means (averaged over time) using

the procedure PROC RANK in SAS. Tukey's Studentised Range test was employed

for pairwise comparisons.

Results

The demographic characteristics of the enrolled subjects are shown in Table

1. In total, 28 of the 30 subjects completed the study, of whom 20 completed

all scheduled visits and eight subjects missed one scheduled visit. One

subject discontinued from the study owing to an adverse event unrelated to

treatment and a second subject discontinued after missing two visits. All

subjects were included in the analysis.

Maximum scores at sites treated with eflornithine HCl 13.9% cream were

greater than for vehicle-treated sites and less than at sodium lauryl

sulphate-treated sites (Table 3). Cumulative irritation scores were 701 at

sites treated with eflornithine 13.9% cream, 396 at vehicle cream-treated

sites and 1625 at sodium lauryl sulphate-treated sites, out of a possible

maximum of 2016 (Table 4). Tukey's Studentised Range test and Friedman's

test showed that the mean scores for the three treatments were significantly

different from each other (p < 0.001) (Table 4).

One subject reported chest tightness and dizziness during the cumulative

irritation study; these events were considered unrelated to the study

treatments. One subject also complained of itchy dry skin unrelated to patch

sites. No other adverse events were reported.

Phototoxicity Study

Subjects and Methods

In total, 25 subjects were enrolled in an open-label, single-centre,

within-subject vehicle-controlled study to evaluate the phototoxicity

potential of eflornithine HCl 13.9% cream and its vehicle alone. The study

consisted of a single application of each study material made to stripped

skin sites followed by irradiation with ultraviolet light. Skin responses

were assessed during the following two days[11, 14]. Healthy subjects were

enrolled in the study based on the same criteria as before. Additionally,

subjects with a recent tan, sunburn or cataracts, or taking medications

suspected of causing photobiological reactions (e.g. tetracyclines and

thiazides), were excluded.

Three sites on the back of each subject were prepared by stripping the skin

with cellophane tape. The skin was stripped to the glistening layer, or a

maximum of 15 repetitions of the stripping process. Eflornithine HCl 13.9%

cream (0.2 g) was applied to one 2.54 cm2 patch of stripped skin (i.e. 80 mg

eflornithine HCl 13.9% cream per square centimetre) and vehicle cream alone

was applied to a second patch, while the third site was left untreated. The

creams were allowed to dry and a portion of each treated site was covered

with an opaque material. All three sites were then exposed to filtered UVA

light for an exposure time equal to 10 times the minimal erythema dose

(MED), followed by an additional 0.5 MED of unfiltered UVA and UVB light,

from a xenon lamp solar simulator. The MED of each subject had been

determined previously using a 1000 W Oriel Solar Simulator (peak

transmission 320-4000 nm, UVA output 45.5 mW/cm2, UVB output 6.0 mW/cm2).

All sites were examined for signs of skin reaction using the same five-point

ordinal scale as before, immediately after irradiation and 20 minutes, 3

hours, 24 hours and 48 hours thereafter. Adverse events were recorded for

the duration of the study for all subjects enrolled.

Results

The demographic characteristics of the enrolled subjects are shown in Table

1. All 25 subjects completed the study. One subject missed the three-hour

and 24-hour evaluations but was not excluded from the analyses.

Following a single treatment with eflornithine HCl 13.9% cream and

subsequent irradiation, 10 of 25 sites (40%) showed no sign of reaction

(Table 5). The remaining 15 irradiated sites treated with eflornithine 13.9%

cream had maximum scores of 1 (slight erythema), all but one falling to 0

within 24 hours. The same pattern of reaction was seen at vehicle

cream-treated and untreated irradiated sites. No sign of reaction was

detected at non-irradiated sites treated with eflornithine HCl 13.9% cream

or vehicle alone (scores of 0). No adverse events were reported during the

phototoxicity study.

Photocontact Allergy Study

Subjects and Methods

In total, 30 subjects were enrolled in an open-label, single-centre,

within-subject vehicle-controlled study to evaluate the photoallergic

potential of eflornithine HCl 13.9% cream and vehicle alone. Subjects were

enrolled using the same criteria as the phototoxicity study.

Twice-weekly during a three-week induction period, eflornithine HCl 13.9%

cream and vehicle alone (0.2 g of each) were applied in duplicate under

occlusive patches to sites 1.8 cm in diameter on the subjects' backs. The

patches were removed 24 hours after application and one of each pair of

duplicate sites, plus an untreated site, were irradiated with 2 MEDs of

unfiltered ultraviolet light (UVA and UVB) using a solar simulator.

Following a two-week no-treatment period, a challenge application of study

materials was made as before, to previously untreated sites. After 24 hours,

one of each of the duplicate treated sites and an untreated site were

irradiated with 10 MEDs of filtered ultraviolet light (UVA).

All sites were examined for signs of skin reaction using the same five-point

ordinal scale as before, five minutes, 20 minutes, 24 hours, 48 hours and 72

hours after irradiation. Adverse events were recorded for the duration of

the study for all subjects enrolled.

Results

The demographic characteristics of the enrolled subjects are shown in Table

1. Of the 30 subjects enrolled, 28 completed the study and were included in

the analysis. Two subjects left the study, of their own volition.

During the induction period, all irradiated sites (treated with eflornithine

HCl 13.9% cream, vehicle-treated and untreated) had at least one score of 1

and there were no scores greater than 1. During induction, most

non-irradiated sites treated with eflornithine HCl 13.9% cream (85.7%) had a

score of 0 throughout, three sites (10.7%) had single scores of 1 and one

site (3.6%) had a single score of 2. During induction at vehicle-treated,

non-irradiated sites, 12 sites (42.9%) had a score of 0 throughout and the

remaining 16 sites (57.1%) had scores of 1 on one or two occasions.

After challenge, there was no sign of reaction at over half of the

irradiated sites (sites treated with eflornithine HCl 13.9%; cream 64.3%;

vehicle-treated 57.1%; untreated 64.3%) and most of the non-irradiated sites

(sites treated with eflornithine HCl 13.9%; cream 85.7%; vehicle-treated

85.7%) (Table 6). The remaining sites had signs of mild erythema five or 20

minutes after challenge, which disappeared within 24 hours.

No serious adverse events were reported in this study. Four adverse events

were reported in three subjects: dry skin at a site treated with

eflornithine HCl 13.9% cream (considered related to study medication),

itching at skin test sites during the third week of study (considered

possibly related to study medication), bronchitis (considered unrelated to

treatment) and stress (considered unrelated to treatment).

Discussion

In these studies, test conditions were created to assess the potential of

eflornithine HCl 13.9% cream to provoke irritant, allergic, photoallergic

and phototoxic dermal reactions. The results provide no evidence to suggest

that either eflornithine HCl 13.9% cream or its vehicle alone induces

phototoxic or photosensitisation skin reactions. In the contact

sensitisation study, the intensity of reaction in most subjects was low and

decreased substantially within 24 hours of challenge. These characteristics

are indicative of irritation as opposed to allergic contact sensitisation.

Under exaggerated conditions of repeated, occluded exposure, eflornithine

HCl 13.9% cream produced signs of dermal irritation in most subjects. The

mean cumulative irritation score for eflornithine HCl 13.9% cream was

significantly greater than for vehicle alone, but significantly less than

for the known irritant sodium lauryl sulphate (0.5%). These findings suggest

that eflornithine HCl 13.9% cream could cause irritation reactions in

clinical use in susceptible individuals or under exaggerated conditions.

Adverse events during exaggerated treatment with eflornithine HCl 13.9%

cream and vehicle alone were generally mild and none was serious. The only

treatment-related adverse events in the four studies (315 subjects in total)

were pruritus (three subjects) and dry skin (one subject) at test sites.

The results of these studies together suggest that eflornithine HCl 13.9%

cream will have a good dermal safety profile in clinical use, with a low

risk of skin irritation, allergic reactions and phototoxicity. These results

complement the findings of efficacy studies that show eflornithine HCl 13.9%

cream to be a highly effective treatment for inhibiting facial hair growth

(manuscript in preparation). The favourable dermal safety profile of

eflornithine HCl 13.9% cream combined with its efficacy in reducing facial

hair growth suggest that eflornithine HCl 13.9% cream offers a significant

breakthrough in the management of unwanted facial hair.

Table 1. Demographic characteristics of subjects enrolled in dermal safety

studies

Study Contact

sensitisation Cumulative

irritation Phototoxicity Photocontact

allergy

Subjects enrolled (No.) 230 30 25 30

Subjects completing (No.) 208 28 25 28

Age (years)

mean 44.9 48.0 39.5 41.4

range 18-87 29-73 22-76 20-73

Gender (% female) 75.2 83.3 88.0 83.3

Race (%)

Black 58.7 36.7 0.0 3.3

White 40.9 63.3 100.0 96.7

Asian/Pacific Islander 0.4 0.0 0.0 0.0

Table 2. Maximum irritation score five minutes and 24 hours after challenge

in a modified Draize skin sensitisation test of eflornithine HCl 13.9% cream

and its vehicle (contact sensitisation study)

Maximum score on the

irritation scale Eflornithine HCl 13.9% cream Vehicle

Five minutes

after challenge 24 hours after

challenge Five minutes

after challenge 24 hours after

challenge

No. % No. % No. % No. %

0 or 1 No sign of reaction

or slight erythema 204 98.1 207 99.5 207 99.5 208 100.0

2 Noticeable

erythema with

slight infiltration 3 1.4 1 0.5 1 0.5 0 0.0

3 Erythema with

marked oedema 0 0.0 0 0.0 0 0.0 0 0.0

4 Erythema with

oedema and

blistering 1 0.5 0 0.0 0 0.0 0 0.0

Total 208 100.0 208 100.0 208 100.0 208 100.0

Table 3. Maximum irritation scores recorded during the cumulative irritation

study: three weeks of daily treatment with eflornithine HCl 13.9% cream,

vehicle alone and 0.5% sodium lauryl sulphate in petrolatum

Maximum score on irritation scale Eflornithine HCl

13.9% cream Vehicle Sodium lauryl

sulphate

No. % No. % No. %

0 No sign of reaction 0 0.0 0 0.0 0 0.0

1 Slight erythema 5 16.7 15 50.0 1 3.3

2 Noticeable erythema with slight infiltration 7 23.3 12 40.0 2 6.7

3 Erythema with marked oedema 1 3.3 2 6.7 0 0.0

4 Erythema with oedema and blistering 17 56.7 1 3.3 27 90.0

Total 30 100.0 30 100.0 30 100.0

Table 4. Total cumulative and mean scores by treatment (n = 30) during the

cumulative irritation study: three weeks of daily treatment with

eflornithine HCl 13.9% cream, vehicle alone and 0.5% sodium lauryl sulphate

in petrolatum

Irritation score Eflornithine HCl

13.9% cream Vehicle Sodium lauryl

sulphate

Cumulative*

Mean? 1.33 0.76 3.09

Tukey's test? B C A

*Sum of all readings for subjects for a given product (maximum score 2016)

?p < 0.001 (Friedman's test)

?Means with different letters are significantly different

Table 5. Maximum irritation scores and scores 48 hours after irradiation

during phototoxicity study with eflornithine HCl 13.9% cream and vehicle

(with and without irradiation) or irradiation alone

Maximum score on

irritation scale Eflornithine HCl 13.9% cream

n (%) Vehicle

n (%) Untreated

n (%)

Irradiated Non-irradiated Irradiated Non-irradiated Irradiated

Max 48 hour Max Max 48 hour Max Max 48 hour

0 No sign of reaction 10 (40) 24 (96) 25 (100) 10 (40) 24 (96) 25 (100) 10

(40) 24 (96)

1 Slight erythema 15 (60) 1 (4) 0 (0) 15 (60) 1 (4) 0 (0) 15 (60) 1 (4)

2 Noticeable erythema

with slight infiltration 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0)

3 Erythema with marked

oedema 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0)

4 Erythema with oedema

and blistering 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0)

Total 25 (100) 25 (100) 25 (100) 25 (100) 25 (100) 25 (100) 25 (100) 25

(100)

Table 6. Irritation scores during photocontact allergy study after treatment

with eflornithine HCl 13.9% cream or vehicle (with and without irradiation)

or irradiation alone: scores up to 20 minutes or 24 hours after irradiation

challenge

Maximum score on

irritation scale Eflornithine HCl 13.9% cream Vehicle Untreated

Irradiated Non-irradiated Irradiated Non-irradiated Irradiated

20 min

n (%) 24 hours

n (%) 20 min

n (%) 24 hours

n (%) 20 min

n (%) 24 hours

n (%) 20 min

n (%) 24 hours

n (%) 20 min

n (%) 24 hours

n (%)

0 No sign of reaction 18 (64.3) 28 (100) 24 (85.7) 28 (100) 16 (57.1) 28

(100) 24 (85.7) 28 (100) 18 (64.3) 28 (100)

1 Slight erythema 10 (35.7) 0 (0) 4 (14.3) 0 (0) 12 (42.9) 0 (0) 4 (14.3) 0

(0) 10 (35.7) 0 (0)

2 Noticeable

erythema with

Sslight infiltration 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0

(0)

3 Erythema with

marked oedema 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0)

4 Erythema with

oedema and

blistering 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0) 0 (0)

Total 28 (100) 28 (100) 28 (100) 28 (100) 28 (100) 28 (100) 28 (100) 28

(100) 28 (100) 28 (100)

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