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NATAP - http://www.natap.org

Trial of TMC114 Administered with Low Dose Ritonavir (RTV) in HIV-1 Infected Treatment Experienced Patients

clinicaltrials.gov

Study TMC114-C214 is a randomized, controlled, open-label trial to compare the efficacy, safety and tolerability of TMC114 boosted with low dose ritonavir (RTV) versus lopinavir (LPV)/RTV in treatment-experienced HIV-1 infected patients.

Primary Outcomes: Change in viral load at 48 weeks.

Secondary Outcomes: Evaluate safety, tolerability and durability of efficacy over 96 weeks.

Expected Total Enrollment: 500

Study start: April 2005; Expected completion: March 2008

Last follow-up: November 2007; Data entry closure: December 2007

Study TMC114-C214 is a randomized, controlled, open-label trial to compare the efficacy, safety and tolerability of TMC114 boosted with low dose ritonavir (RTV) versus lopinavir (LPV)/RTV in treatment-experienced HIV-1 infected patients.

This research study will look at the safety of TMC114 and its effectiveness in reducing the amount of HIV (viral load) in the blood.

People included in this study will have received either Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTIs) or Protease Inhibitors (PIs) or both. Major inclusion and exclusion criteria are listed below.

The duration of the study will be approximately 106 weeks, which includes a 4 to 6 week screening period, 96-week treatment period, and 4-week follow-up period.

Eligibility

Ages Eligible for Study: 18 Years and above, Genders Eligible for Study: Both

Criteria

Inclusion Criteria:

* Patient has documented HIV-1 infection

* Treatment with an Antiretroviral regimen (containing at least 2 NRTIs in combination with at least 1 NNRTI and/or 1 PI) for at least 12 weeks

* Plasma HIV-1 RNA >1000 copies/mL

* General medical condition does not interfere with the assessments and the completion of the trial

Exclusion Criteria:

* Patients for whom an investigational Antiretroviral is part of the current regimen, with the following exceptions if applicable (depending on local regulatory approval); tenofovir, emtricitabine, atazanavir, fosamprenavir

* Previous or current use of lopinavir, enfuvirtide (T-20), tipranavir and TMC114

* Life expectancy of less than 6 months

* Pregnant or breast-feeding

* Females of childbearing potential not willing to use effective non-hormonal birth control methods or not willing to continue practicing these birth control methods for at least 14 days after the end of the treatment period

* Patients with significantly decreased liver function or decompensation, irrespective of liver enzyme levels

* Participation in other investigational trials without prior approval of the sponsor

STUDY SITES

Location and Contact Information

Please refer to this study by ClinicalTrials.gov identifier NCT00110877

M McShane cmcshane@...

Arizona

Body Positive, Inc., Phoenix, Arizona, 85006, United States; Not yet recruiting

Barbara Casimir, BSN, CCRP Ext. 2225

A. Myers, MD, Principal Investigator

Arkansas

Health For Life Clinic, Pllc, Little Rock, Arkansas, 72207, United States; Not yet recruiting

Montgomery bmontgomery@...

Jefferson, MD, Principal Investigator

California

Goodman Clinic, DBA L.A. Gay and Lesbian Center,

Los Angeles, California, 90028, United States;

Not yet recruiting

Bolan, MD, Principal Investigator

East Bay AIDS Center,

Berkeley, California, 94705, United States;

Not yet recruiting

Mandelke

mandelh@...

Borkert, MD, Principal Investigator

AIDS Research Alliance,

West Hollywood, California, 90069, United States;

Not yet recruiting

Grace Gacherja

mvertucci@...

Brown, MD, Principal Investigator

AIDS Healthcare Foundation Research Center,

Los Angeles, California, 90015, United States; Not yet recruiting

Farthing, MD, Principal Investigator

Kaiser Permanente Medical Center,

San Francisco, California, 94115, United States;

Not yet recruiting

W. Fessel, MD, Principal Investigator

Cedars-Sinai Medical Center,

Los Angeles, California, 90048, United States; Not yet recruiting

Gregg Sannes

Hardy, PhD, Principal Investigator

Kaiser Permanente,

Los Angeles, California, 90027, United States;

Not yet recruiting

Guinto, MPH

Marc LaRiviere, MD, Principal Investigator

Tony Mills/ Ruane, MD,

Los Angeles, California, 90069, United States;

Not yet recruiting

Alas Ext. 15

Ruane, MD, Principal Investigator

Living Hope Clinical Foundation,

Long Beach, California, 90813, United States;

Not yet recruiting

o Yolo

ryolo@...

Stefan Schneider, MD, Principal Investigator

San Francisco VA Medical Center,

San Francisco, California, 94121, United States;

Not yet recruiting

Harry Lampiris, MD, Principal Investigator

Colorado

University of Colorado,

Denver, Colorado, 80262, United States;

Not yet recruiting

Suzanne Fiorillo

suzanne.fiorillo@...

B. , MD, Principal Investigator

District of Columbia

Capital Medical Associates,

Washington, District of Columbia, 20036, United States; Not yet recruiting

Seymour

alex@...

Bruce S. Rashbaum, MD, Principal Investigator

Washington Univ. Medical Center,

Washington, District of Columbia, 20037, United States;

Not yet recruiting

Bisby

nbisby@...

Afsoon , MD, Principal Investigator

Whitman- Clinic, Washington,

District of Columbia, 20009, United States;

Not yet recruiting

Christiane Geisler

Kunthavi Sathasivam, MD, Principal Investigator

Florida

IDC Research Initiative,

Altamonte Springs, Florida, 32701, United States;

Not yet recruiting

Charmaine Stiles

Ext. 3102 cstiles@...

Edwin DeJesus, MD, Principal Investigator

University of Miami School of Medicine,

Miami, Florida, 33136, United States;

Not yet recruiting

Kaszubski, RN ckaszubs@...

Dushyantha T. Jayaweera, MD, Principal Investigator

Clin. Res. Ctr. at Tampa General Hospital,

Tampa, Florida, 33606, United States;

Not yet recruiting

Mable Chow Ext. 6460 mable_chow@...

P. Nadler, MD, Principal Investigator

St. ph's Comprehensive Research Iniitiative,

Tampa, Florida, 33611, United States;

Not yet recruiting

Ext. 228 jennifer.bailey@...

Dorece G. Norris, MD, Principal Investigator

Treasure Coast Infectious Disease Consultants,

Vero Beach, Florida, 32960, United States; Not yet recruiting

Jeff Mieras

Gerald Pierone, MD, Principal Investigator

Richmond, MD,

Fort Lauderdale, Florida, 33316, United States;

Not yet recruiting

Richmond, MD, Principal Investigator

Health Positive, Safety Harbor, Florida, 34695, United States;

Not yet recruiting

Ross

Barry M. Rodwick, MD, Principal Investigator

HIV Clinical Research, Fort Lauderdale, Florida, 33311, United States; Not yet recruiting

Yontif Ext. 224

hyontif@...

G. Sension, MD, Principal Investigator

Steinhart Medical Associates, Miami, Florida, 33133, United States;

Not yet recruiting

Amy Sue Liebmann Ext. 232

aliebmann@...

Corklin R. Steinhart, MD, Principal Investigator

Infectious Disease Research Institute, Inc.,

Tampa, Florida, 33614, United States;

Not yet recruiting

Kalliope Halkias

kdhalkias@...

Bienvenido G. Yangco, MD, Principal Investigator

Georgia

Atlanta Infectious Disease Group, PC,

Atlanta, Georgia, 30309, United States;

Not yet recruiting

Stadtlander

Philip S. Brachman, MD, Principal Investigator

Infectious Disease Specialists of Atlanta,

Decatur, Georgia, 30033, United States;

Not yet recruiting

Maclure

Robin Dretler, MD, Principal Investigator

Mercer University School of Medicine,

Macon, Georgia, 31201, United States;

Not yet recruiting

Harold Katner, MD, Principal Investigator

Atlanta Specialty Research,

Atlanta, Georgia, 30342, United States;

Not yet recruiting

L. Usherwood, MMSc, PA-C jusherwood@...

I. Marlowe, MD, Principal Investigator

AIDS Research Consortium of Atlanta, Inc,

Atlanta, Georgia, 20208, United States;

Not yet recruiting

To Be Determined

A. , MD, Principal Investigator

Illinois

Northstar Medical Center,

Chicago, Illinois, 60657, United States;

Recruiting

Elonia

Berger, MD, Principal Investigator

Northwestern University Feinberg School of Medicine,

Chicago, Illinois, 60611, United States;

Not yet recruiting

Baiba Berzins

Palella, MD, Principal Investigator

Kentucky

University of Kentucky School of Medicine,

Lexington, Kentucky, 40536, United States;

Not yet recruiting

Plummer

slplum2@...

N. Greenberg, MD, Principal Investigator

Massachusetts

Community Research Initiative of New England,

Boston, Massachusetts, 02215, United States;

Not yet recruiting

Anne Habel Ext. 225

ahabel@...

Amy Colson, MD, Principal Investigator

Community Research Initiative of New England,

Springfield, Massachusetts, 01107, United States;

Not yet recruiting

Margarita Canuel, RN

mcanuel@...

Anne B. , MD, Principal Investigator

Michigan

Benson, DO, Berkley, Michigan, 48072, United States;

Not yet recruiting

Dorothy Dempster dorothydempster@...

Benson, DO, Principal Investigator

Minnesota

Clinic 42, Minneapolis, Minnesota, 55404, United States;

Not yet recruiting

Vern Appleby

vfappleby@...

S. Rhame, MD, Principal Investigator

New Jersey

University Hospital,

Camden, New Jersey, 08103, United States;

Not yet recruiting

Deborah Goraj Ext. 3518

Baxter, MD, Principal Investigator

VA NJ Healthcare System,

East Orange, New Jersey, 07018, United States;

Not yet recruiting

Latorre, RN Ext. 2146

Eng, MD, Principal Investigator

Saint 's Medical Center,

Newark, New Jersey, 07102, United States;

Not yet recruiting

Fallon

jimf@...

M. , MD, Principal Investigator

New York

NBHN, Bronx, New York, 10461, United States;

Not yet recruiting

Agelo Sedg, RN

Leider, MD, Principal Investigator

North Carolina

Duke University Medical Center, Durham, North Carolina, 27710, United States; Not yet recruiting

ta Giner giner001@...

B. Hicks, MD, Principal Investigator

Jemsek Clinic,

Huntersville, North Carolina, 28078, United States;

Not yet recruiting

Harper eharper@...

ph G. Jemsek, MD, Principal Investigator

Wake Forest University Health Sciences,

Winston Salem, North Carolina, 27157, United States;

Not yet recruiting

Hauser

smhauser@...

Aimee Wilkin, MD, Principal Investigator

Ohio

University of Cincinnati,

Cincinnati, Ohio, 45267, United States;

Not yet recruiting

Tamar Canaan

Judith Feinberg, MD, Principal Investigator

Cleveland Clinic Foundation,

Cleveland, Ohio, 44195, United States;

Not yet recruiting

Colleen Workman

Alan Taege, MD, Principal Investigator

Oregon

The Research & Education Group,

Portland, Oregon, 97209, United States;

Not yet recruiting

Norma ez

Sampson, MD, Principal Investigator

Pennsylvania

Philadelphia FIGHT,

Philadelphia, Pennsylvania, 19107, United States;

Not yet recruiting

Barbara A. Gallagher, RN

Karam Mounzer, MD, Principal Investigator

The Drexel University College of Medicine,

Philadelphia, Pennsylvania, 19102, United States;

Not yet recruiting

Regina , RN, MSN regina.anthony@...

R. Short, MD, Principal Investigator

South Carolina

The Burnside Clinic,

Columbia, South Carolina, 29206, United States;

Not yet recruiting

Felder, III

rick@...

Alfred F. Burnside, Jr., MD, Principal Investigator

Tennessee

Vanderbilt Aids Clinical Trial Center,

Nashville, Tennessee, 37203, United States;

Not yet recruiting

Janet Nicotera

Haas, MD, Principal Investigator

Texas

University of Texas Houston Medical School,

Houston, Texas, 77030, United States;

Not yet recruiting

Berta

Ben J. Barnett, MD, Principal Investigator

Professional Quality Research, Inc.,

Austin, Texas, 78756, United States;

Not yet recruiting

Mol

tracy@...

Jack Bissett, MD, Principal Investigator

North Texas Center for Aids and Clinical Research,

Dallas, Texas, 75208, United States;

Not yet recruiting

Brand, MD, Principal Investigator

Central Texas Clinical Research,

Austin, Texas, 78705, United States;

Not yet recruiting

Tom Brinson tbrinson@...

Brinson, MD, Principal Investigator

University of Texas Medical Branch,

Galveston, Texas, 77555, United States;

Not yet recruiting

Cheryl Mogridge

clmogrid@...

A. O'Brien, MD, Principal Investigator

Special Health Resources for Texas Incorporated,

Longview, Texas, 75601, United States;

Not yet recruiting

Lawrence

Anita Scribner, MD, Principal Investigator

Montrose Clinic, Houston, Texas, 77098, United States;

Not yet recruiting

Mark Mall

mmall@...

R Schrader, MD, Principal Investigator

Virginia

Hampton Roads Medical Specialists,

Hampton, Virginia, 23666, United States;

Not yet recruiting

Katy Schwarzenberg Ext. 15 hrms21@...

Green, MD, Principal Investigator

Washington

Swedish Medical Center,

Seattle, Washington, 98122, United States;

Not yet recruiting

Algren

Shalit, MD, Principal Investigator

Wisconsin

Froedtert & Medical College Froedtert East Clinic Bldg., Milwaukee, Wisconsin, 53226, United States;

Not yet recruiting

Mandy Kastner

, MD, Principal Investigator

Puerto Rico

Clinical Research Puerto Rico, Inc.,

San , 00909-1711, Puerto Rico;

Not yet recruiting

Ana L. Campos, RN, MBA/HCM

Morales , MD, Principal Investigator

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